Panel Discussion: Debating the Relevance of GPCR Dimers and Whether Signaling through GPCR Heterodimers is Pharmacologically Relevant

Time: 9:00 am
day: Day Two


  • We acknowledge dimerization occurs, but what is the pharmacological relevance?
  • Can you selectively target GPCR heterodimers using ligands that bind both dimers or monomers?
  • How can we leverage experimental data on dimerization, computationally?