What Can You Expect at the Premier GPCR Forum in 2026?

With GPCR investment surging and multi-billion-dollar deals redefining the competitive landscape, the race is on to unlock new receptors and modalities.

The 5th GPCR-Targeted Drug Discovery Summit delivers:

  • Exclusive perspectives
  • Never-seen-before data
  • Practical strategies from teams leading the field

Gain actionable insights to accelerate GPCR therapeutics discovery and stay ahead of industry momentum.

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Top Sessions for 2026:

Harnessing AI & ML for Smarter GPCR Drug Discovery

Insights from: Nabla Bio,Biagon, Eli Lilly, Iambic Therapeutics and more

Advancing Next-Generation Antibody and Peptide Approaches

Insights from: Skymab Biotherapeutics, Confo Therapeutics, GSK more

Optimizing Translational Strategies for Clinical Impact

Insights from: Tectonic Therapeutics, Atai Life Sciences, Domain Therapeutics and more

Interrogating the Functional Significance of GPCR Signaling

Insights from: InterAx Biotech, Northeastern University and more

Explore The Full Event Guide

  • 80+ Attendees
  • 25+ World-Class Speakers
  • 21+ Data-Driven Presentations
  • 7+ Hours of Networking
  • 1 AI & ML Focus Day
69612 - 5th GPCRs-Targeted Drug Discovery Summit

Attending Companies Include

explore the agenda
Explore the Agenda

Hear the latest industry breakthroughs and gain exclusive insights during our packed agenda, interactive roundtables, and panel discussions.

Join Biopharma Experts
Join Biopharma Experts

Be part of the hottest conversations with like-minded attendees spanning all stages of drug discovery and make critical connections during our dedicated networking sessions

Partner With Us
Partner With Us

Position yourself alongside other leading solution providers to ensure your brand is at the heart of biopharma deals.